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| Preface | |
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| Solid-Phase Synthesis: Basic Principles | |
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| Solid Supports | |
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| Linkers | |
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| Reaction Monitoring in Solid-Phase Synthesis | |
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| Purity and Yield Determination in Solid-Phase Synthesis | |
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| References | |
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| Solid-Phase Synthesis: Oligomeric Molecules | |
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| Peptides | |
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| Oligonucleotides | |
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| Oligosaccharides | |
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| References | |
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| Solid-Phase Synthesis: Small Organic Molecules | |
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| Small Organic Molecules on Solid Phase: Target Selection and Solution Studies | |
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| Small Organic Molecules on Solid Phase: Solid-Phase Synthesis | |
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| Small Organic Molecules on Solid Phase: From Solid-Phase Synthesis to Synthetic Organic Libraries | |
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| An Example: Solid-Phase Synthesis of 1H-[2]Pyrindinones | |
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| Solid-Phase Synthetic Strategies: Selected Examples | |
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| References | |
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| Combinatorial Technologies: Basic Principles | |
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| Combinatorial Technologies | |
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| Combinatorial Libraries | |
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| References | |
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| Synthetic Organic Libraries: Library Design and Properties | |
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| Primary Libraries: Shooting in the Dark? | |
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| Focused Libraries: High-Throughput Structure-Activity Relationships | |
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| Biased-Targeted Libraries: Information-Rich Primary Libraries | |
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| Library Design via Computational Tools | |
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| References | |
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| Synthetic Organic Libraries: Solid-Phase Discrete Libraries | |
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| Synthesis of Solid-Phase Discrete Libraries | |
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| Structure Determination, Quality Control, and Purification of Solid-Phase Discrete Libraries | |
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| Examples of Solid-Phase Discrete Library Synthesis | |
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| New Trends in Solid-Phase Discrete Library Synthesis | |
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| References | |
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| Synthetic Organic Libraries: Solid-Phase Pool Libraries | |
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| Synthesis of Solid-Phase Pool Libraries | |
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| Direct Structure Determination of Positives from Solid-Phase Pool Libraries | |
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| Deconvolution Methods for Solid-Phase Pool Libraries | |
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| Encoding Methods for Solid-Phase Pool Libraries | |
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| New Trends in Solid-Phase Pool Libraries | |
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| References | |
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| Synthetic Organic Libraries: Solution-Phase Libraries | |
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| Solution- Versus Solid-Phase Synthetic Libraries: Which Ones to Use? | |
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| Solution-Phase Discrete Libraries | |
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| Purification of Solution-Phase Library Intermediates and Final Compounds: Liquid-Liquid and Solid-Phase Extraction Systems | |
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| Solid-Phase Assisted Solution-Phase Library Synthesis and Purification | |
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| Soluble Supports in Solution-Phase Combinatorial Synthesis | |
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| New Trends in Solution-Phase Combinatorial Synthesis | |
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| References | |
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| Applications of Synthetic Libraries | |
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| Pharmaceutical Applications | |
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| Agrochemical and Food-Related Applications | |
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| Applications to Combinatorial Reaction Optimization | |
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| Applications to Catalysis | |
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| Applications to Molecular Recognition | |
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| References | |
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| Biosynthetic Combinatorial Libraries | |
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| Biosynthetic Polypetide Libraries | |
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| Biosynthetic Oligonucleotide Libraries | |
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| Combinatorial Biosynthesis of Natural Products | |
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| Combinatorial Biocatalysis | |
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| References | |
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| Materials and Polymeric Combinatorial Libraries | |
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| Synthesis of Materials Science Libraries | |
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| Characterization and Screening of Materials Science Libraries | |
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| Polymeric Combinatorial Libraries | |
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| References | |
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| Index | |